cannabinoid receptor type 1 (CB1) and type 2 (CB2)

April 28, 2021

WIN55,212-2, a Dual Modulator of Cannabinoid Receptors and G Protein-Coupled Inward Rectifier Potassium Channels

Abstract The coupling of cannabinoid receptors, CB1 and CB2, to G protein-coupled inward rectifier potassium channels, GIRK1 and GIRK2, modulates…

July 17, 2020

Targeting Cannabinoid Receptors: Current Status and Prospects of Natural Products

Abstract Cannabinoid receptors (CB1 and CB2), as part of the endocannabinoid system, play a critical role in numerous human physiological…

August 29, 2019

Design and development of stapled transmembrane peptides that disrupt the activity of G-protein–coupled receptor oligomers

Abstract Membrane proteins can associate into larger complexes. Examples include receptor tyrosine complexes, ion channels, transporters, and G protein–coupled receptors…